平安! 发表于 2011-11-9 19:57 2 M) ?' g3 D' b6 U
Pazopanib (100 mg/kg/day free base equivalent) 6 H+ f9 ~! [* N5 E0 g
这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。
" Z( c' i" {# T2 E& ~8 o2 p搜索了一下,原料一大堆。7 X: N; F: l% j1 Y3 q# |; R8 O5 H
, X) {# W) F& T+ D对不起!100mg/kg是用于移植瘤的,我弄错了。3 T( F- [* {- K: Q* q
9 d F& F6 V4 z- h3 `- b1 D4 V以下是正版说明书的推荐用量。) o7 F+ \9 H2 B6 J4 e% F
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--------------------- DOSAGE AND ADMINISTRATION ----------------
: W3 v2 N w" w5 K6 k* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1) ( V: w, g* |% f
* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) 6 T* K. E/ t$ A6 k* B( ?
---------------------DOSAGE FORMS AND STRENGTHS --------------' p" w5 x% p' s# D. n5 D
200 mg tablets. (3)
% k& |* H7 k0 ]& @2 M/ P- l- c/ J-------------------------------CONTRAINDICATIONS------------------------ |